5th International Symposium on Pharmaceutical Chemistry

September 5-7, Istanbul-TURKEY

e-mail: ispc5@hacettepe.edu.tr

  

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PROGRAMME

 

September 4, 2007 TUESDAY

19.30

WELCOME COCKTAIL

Hotel Sheraton-Istanbul Maslak – Sky Light Ball Room

 

September 5, 2007 WEDNESDAY (GALAXY III HALL)

09.30-10.00

OPENING CEREMONY

10.00-10.45

Morning – 1st Session

Chair Persons

Prof. Shizuo Yamada

10.00-10.45

Richard A. Glennon (Virginia Commonwealth University-USA)

Drug Discrimination: Application to Medicinal Chemistry

10.45-11.00

COFFEE BREAK

11.00-12.30

Morning – 2nd Session

Chair Persons:

Prof. Richard F. Borch

Prof. Mevlüt Ertan

11.00-11.45

Giuseppe Campiani (Siena University-Italy)

Development of the Third Generation Non-Nucleoside HIV-1 RT Inhibitors and Design of Potential HCV Antivirals by Selective Targeting HCV NS3 Helicase

11.45-12.30

David C. K. Chu (The University of Georgia-USA)

Preclinical and Clinical Studies of Clevudine (L-FMAU)as Potent Antiviral Agents Against Chronic Hepatitis B Virus

12.30-13.30

LUNCH

13.30-14.30

POSTER PRESENTATIONS (GALAXY II HALL)

14.30-16.00

Afternoon – 1st Session

Chair Persons:

Prof. Hermann Waetzig

Prof. Malgorzata Dukat

14.30-15.15

Margaret O. James (University of Florida-USA)

Inhibition of Sulfotransferases

15.15-16.00

Jiang Zheng (Seattle Children’s Hospital Research Institute-USA)

Metabolism and Bioactivation of Styrene

16.00-16.30

Nazlı Böke (Ege University-Turkey)

Essential Fatty Acid Components and Antioxidant Activities of Eight Cephalaria Species From Southwestern Anatolia

16.30-17.00

COFFEE BREAK

 

September 6, 2007 THURSDAY (GALAXY III HALL)

09.00-10.30

Morning – 1st Session

Chair Persons:

Prof. Margaret O. James

Prof. Giuseppe Campiani

09.00-09.45

Shizuo Yamada (University of Shizuoka-Japan)
In Vivo Analysis of Drug-Receptor Binding Characteristics in Drug Discovery

09.45-10.30

Prof. Caterina Fattorusso (NatSynDrugs-Italy)

Exploiting Protein Fluctuations at the Active Site Gorge of Cholinesterases: Further Optimization of the Design Strategy to Extremely Potent Multiple Binding Site Inhibitors

10.30-11.00

COFFEE BREAK

11.00-12.30

Morning – 2nd Session

Chair Persons:

Prof. Ahmed Mehanna

Prof. Hülya Akgün

11.00-11.45

Laurence Hurley (Arizona University-USA)

A New Strategy for Modulation of Gene Expression by Small Molecules

11.45-12.30

Ongun Onaran (Ankara University-Turkey)

Exploring Allosteric Coupling in G Protein Alpha Subunit by Using Evolutionary, Statistical Ensemble and Dynamycal Approches

12.30-13.30

LUNCH

13.30-14.30

POSTER PRESENTATIONS (GALAXY II HALL)

14.30-15.45

Afternoon – 1st Session

Chair Persons:

Prof. David C. K. Chu

Prof. Dilek Erol

14.30-15.15

Mahmoud H. el Kouni (University of Alabama at Birmingham-USA)

6-Benzylthioinosines: Subversive Substrates of Toxoplasma gondii Adenosine Kinase 

15.15-15.45

Yusuf Mohammad Ali Al-Hiari (University of Jordan-Jordan)

Synthesis and Antibacterial Properties of New 8-Nitro fluoroquinolone Derivatives

15.45-16.15

COFFEE BREAK

15.45-17.15

Afternoon – 2nd Session

Chair Persons:

Prof. Sevim Dalkara

Prof. Hossein Loghmani-Khouzani

16.15-16.45

Dr. Mohamed Gomaa (Cardiff University-UK)

Design And Synthesis Of Some Cyp26 Inhibitors As Indirect Differentiating Agents For Prostate And Breast Cancer

16.45-17.15

Dr. Stefania Butini (NatSynDrugs-Italy)

Development of Potent Atypical Antipsychotics Based on a Novel Neurochemical Approach

20.00-24.00

GALA DINNER

LUFER BOAT – BOSPHORUS CRUISE (Please contact with Organizing Secretariat)

 

 September 7, 2007 FRIDAY (GALAXY III HALL)

09.00-10.30

Morning – 1st Session

Chair Persons:

Prof. Caterina Fattorusso

Prof. Laurence Hurley

09.00-09.45

Richard F. Borch (Purdue University-USA)

Novel Approaches to the Intracellular Delivery of Phosphotyrosine Peptidomimetics and Other Bioactive Phosphates

09.45-10.30

Mohamed Abdel Hamid Ismail (Ain Shams University-Egypt)

Hypotheses Generations for ACEIs, Ang-II Antagonists &  α-1 Adrenoceptor Antagonists for Virtual Screening of Designed Respective Selective anti-hypertensive Agents

10.30-11.00

COFFEE BREAK

11.00-12.30

Morning – 2nd Session

Chair Persons:

Prof. Mahmoud H. el Kouni

Prof. Jiang Zheng

11.00-11.45

Hermann Waetzig (Carola Wilhelmina Technical University-Germany)

Towards Precise and Validated Methods in Pharmaceutical Analysis

11.45-12.30

Satomi Onoue (University of Shizuoka-Japan)

Long-Lasting Analogues and Drug Delivery Systems of Vasoactive Intestinal Peptide for the Treatment of  COPD

12.30-13.00

CLOSING CEREMONY